Fatty alcohol esters
Medchemexpress LLC Histrelin acetate | 220810-26-4 | 99.9% | 1323.50 (free base) | 10 MG
Histrelin acetate is a GnRH analogue and a GnRH Receptor agonist. It increases serum luteinising hormone (LH), follicle stimulating hormone (FSH), and testosterone levels. It can be used in the research of prostate cancer and endometriosis.
- Stimulates the release of vasopressin (VP) and oxytocin (OT) from isolated rat hypothalamo-neurohypophysial explants.
- Rescues circulating LH concentrations in Csfmop/Csfmop mice.
- Reduces the number of endometrial glands, atrophying the stroma in rabbits.
Medchemexpress LLC Glp-1(7-37) acetate | 1450806-98-0 | 99.59% | 3355.67 (free base) | 10 MG
GLP-1(7-37) acetate is an intestinal insulinotropic hormone that augments glucose induced insulin secretion and is for research use only.
- Augments glucose induced insulin secretion
- Solid appearance
- White to off-white color
- Sequence: His-Ala-Glu-Gly-Thr-Phe-Thr-Ser-Asp-Val-Ser-Ser-Tyr-Leu-Glu-Gly-Gln-Ala-Ala-Lys-Glu-Phe-Ile-Ala-Trp-Leu-Val-Lys-Gly-Gr-Gly
- Soluble in H2O: 50 mg/mL (ultrasonic and adjust pH to 1 with HCl)
- Soluble in PBS: 2 mg/mL (clear solution; need ultrasonic)
Medchemexpress LLC Bradykinin acetate | 6846-03-3 | 99.6% | 1060.21 | 10 MG
Bradykinin acetate is a potent endothelium-dependent vasodilator known for its ability to lower blood pressure. It is involved in inducing contraction of bronchial and intestinal non-vascular smooth muscle, increasing vascular permeability, and participating in pain mechanisms. This compound is suitable for various research applications, including studies on its role in cardiovascular function, inflammation, and cellular signaling pathways.
- Effective endothelium-dependent vasodilator
- Lowers blood pressure
- Induces contraction of bronchial and intestinal non-vascular smooth muscle
- Increases vascular permeability
- Participates in pain mechanisms
- Stable for 2 years at -80°C as powder
- Stable for 6 months at -80°C in solvent under sealed, moisture-free conditions
Medchemexpress LLC Ulipristal acetate | 126784-99-4 | 475.62 | 100 MG
Ulipristal acetate (CDB-2914) is an orally active, selective progesterone receptor modulator (SPRM). It stimulates the autophagic response selectively in leiomyoma cells and has potential for treating benign gynecological conditions like uterine myoma.
- Orally active, selective progesterone receptor modulator
- Stimulates autophagy in leiomyoma cells
- Potential for treating benign gynecological conditions, such as uterine myoma
- Blocks activin A modulation of fibronectin and vascular endothelial growth factor A (VEGF-A) mRNA expression
- Possesses significant antiprogestational activity in vivo
- Decreases incidences of fibroadenomas and adenocarcinomas in the mammary gland
Medchemexpress LLC Retinyl acetate | 127-47-9 | MFCD00019413 | 328.49 | 50 MG
Retinyl acetate is a synthetic acetate ester derived from retinol, demonstrating potential antineoplastic and chemopreventive activities. It has been shown to inhibit the proliferation of tumor cells and is suitable for various in vitro and in vivo studies.
- Inhibits proliferation of tumor cells, such as melanoma cell lines B16 and S91
- Inhibits DMBA-induced mammary carcinogenesis in Sprague-Dawley rats
- Appears as a solid, off-white to light yellow in color
- Soluble in DMSO and corn oil for experimental applications
Medchemexpress LLC α-Amyrin acetate | 863-76-3 | 1 MG
α-Amyrin acetate is a pentacyclic triterpenoid compound with oral activity. It inhibits cancer cell proliferation, induces apoptosis, and reduces blood glucose levels. This compound is used for research in cancer and metabolic diseases, such as breast cancer and diabetes.
- Inhibits proliferation and colony formation in MDA-MB-231 cells.
- Induces apoptosis and increases caspase-3 activity in MDA-MB-231 cells.
- Promotes cleavage of Poly polymerase, increases E-cadherin, and inhibits vimentin and phosphorylated extracellular signal-regulated activation in MDA-MB-231 cells.
- Reduces blood glucose levels in diabetic rats.
Medchemexpress LLC JMV 449 acetate | 141863-45-8 | 99.7% | 807.03 | 1 MG
JMV 449 acetate is a potent neurotensin receptor agonist. It exhibits an IC50 of 0.15 nM for inhibiting 125I-neurotensin binding to neonatal mouse brain and an EC50 of 1.9 nM in contracting the guinea-pig ileum. This product also demonstrates highly potent and long-lasting hypothermic and analgesic effects in mice.
- Potent neurotensin receptor agonist
- IC50 of 0.15 nM for inhibition of 125I-neurotensin binding
- EC50 of 1.9 nM in contracting guinea-pig ileum
- Highly potent and long-lasting hypothermic effects
- Highly potent and long-lasting analgesic effects in mice
- White to off-white solid appearance
- Soluble in H2O at 100 mg/mL (requires ultrasonic)
Medchemexpress LLC DALDA (acetate) | 99.8% | 671.79 | 10 MG
DALDA acetate is a potent and highly selective μ-opioid receptor agonist with a Kᵢ of 1.69 nM. It exhibits antinociceptive and respiratory effects. This compound carries a net positive charge (3+) at physiological pH, making it hydrophilic and more polar than morphine.
- Potent and highly selective μ-opioid receptor agonist
- Kᵢ of 1.69 nM
- Exhibits antinociceptive effects
- Exhibits respiratory effects
- Carries a net positive charge (3+) at physiological pH
- More polar than morphine
Medchemexpress LLC BIMAX1 (acetate) | 96.1% | 3542.03 (free base) | 10 MG
BIMAX1 acetate is a tool peptide used to investigate the interaction of RBBP4 with importin β1 and its effects on the nuclear import pathway. It can be employed to study RBBP4's role in regulating nuclear import efficiency and cellular senescence.
- Utilized for investigating RBBP4 and importin β1 interactions
- Helps study nuclear import efficiency
- Can be used to research cellular senescence
- Appears as a white to off-white solid
TARGETMOL CHEMICALS INC Terlipressin Acetate 25MG
Also available in 5 mg, 10 mg, 50 mg, 100 mg, 200 mg and bulk. Please contact Fisher for quotes. Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on oxygen and glucose deprivation/re-oxygenation (OGD/R)-induced damage in intestinal epithelial cells (IEC-6).Terlipressin acetate exerts anti-inflammatory and anti-oxidative effects. Terlipressin acetate has the potential for hepatorenal syndrome and norepinephrine-resistant septic shock research. Purity 99.69%
TARGETMOL CHEMICALS INC CASPOFUNGIN ACETATE 25MG
Also available in 5 mg 10 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Caspofungin Acetate (MK 0991) is the acetate salt of an antimycotic echinocandin lipopeptide semisynthetically derived from a fermentation product of the fungus Glarea lozoyensis. This agent is active against Aspergillus and Candida species. purity: 99%
Medchemexpress LLC Cetrorelix Acetate | 145672-81-7 | 98.25% | 1491.09 | 100 MG
Cetrorelix Acetate is a potent gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM. It is also known as SB-75 acetate. This compound is used in research related to neurological diseases and endocrinology, and has shown antiproliferative effects on cell lines.
- Potent GnRH receptor antagonist
- Inhibits growth of ES-2 cell line
- Applicable in neurological disease research
- Applicable in endocrinology research
Medchemexpress LLC Linaclotide (acetate) | 851199-60-5 | 98.6% | 1586.79 | 50 MG
Linaclotide acetate is a potent and selective guanylate cyclase C agonist; developed for the treatment of constipation-predominant irritable bowel syndrome (IBS-C) and chronic constipation.
- Potent and selective guanylate cyclase C agonist.
- Developed for the treatment of constipation-predominant irritable bowel syndrome (IBS-C).
- Developed for the treatment of chronic constipation.
Medchemexpress LLC Bradykinin acetate | 6846-03-3 | 99.58% | 1060.21 (free base) | 50 MG
Bradykinin acetate | 6846-03-3 | 99.58% | 1060.21 (free base) | 50 MG
Medchemexpress LLC Orbofiban acetate | 163250-91-7 | 98.1% | 421.45 g/mol | C19H27N5O6 | 100 MG
Orbofiban acetate is an orally active platelet GPIIb/IIIa antagonist used in research to inhibit platelet aggregation. It is provided as a solid or as a DMSO solution and intended for in vitro and preclinical studies.
- Orally active platelet GPIIb/IIIa antagonist that inhibits platelet aggregation.
- High purity (approximately 98.1%).
- Molecular formula C19H27N5O6; molecular weight 421.45 g/mol.
- Available as solid (5-500 mg) and as a 10 mM solution in DMSO.
- Soluble in DMSO (≈150 mg/mL) with warming and sonication.
- Storage: solid at 4°C under inert atmosphere; solutions at -80°C (6 months) or -20°C (1 month).
- For research use only; not for human or clinical use.